For general information only. Not a substitute for professional medical advice.
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Educational Medication GuidePrescription OnlyClass: Antimalarial, DMARD

Hydroxychloroquine

Generic Name: Hydroxychloroquine

Common Brand Names: Plaquenil
Dosage Form:Tablet
Route:Oral
Pregnancy Category:C
Last Reviewed:9/21/2026

Uses & Medical Indications

Malaria, rheumatoid arthritis, lupus

Medical Conditions Treated:

RA, SLE

Work Mechanism & Pharmacology

How It Works

Patient Overview of Work Mechanism

Hydroxychloroquine works at the cellular level to correct underlying biochemical imbalances, reduce clinical symptoms, and support overall health.

Clinical Mechanism of Action (MoA)

Hydroxychloroquine exerts targeted therapeutic activity by interacting with specific cellular receptors, enzymatic pathways, or biological signaling cascades to relieve symptoms and restore physiological balance.

Primary TargetHydroxychloroquine sulfate
Therapeutic FamilyAntirheumatic
Administration RouteOral

Dosage & Administration Guidelines

Adult Dosage

200-400 mg daily

Pediatric Dosage

Max 6.5 mg/kg/day

Elderly / Geriatric Considerations

Same as adult

Maximum Dose Limit

400 mg/day

Renal Impairment:

N/A

Hepatic Impairment:

Use with caution

Side Effects & Safety Warnings

Common Side Effects

Nausea, diarrhea, abdominal pain

Serious Adverse Reactions

Retinopathy, QT prolongation, cardiomyopathy

Contraindications:

Retinal or visual field changes

Important Warnings & Precautions:

Irreversible retinal damage can occur

Interactions (Drugs, Food & Alcohol)

Drug-Drug Interactions:

Digoxin, antacids, QT prolonging drugs

Food & Dietary Interactions:

Take with food or milk

Alcohol Interaction Warning:

N/A

Pregnancy & Breastfeeding Safety

Pregnancy Safety

Used in pregnancy for lupus/RA

Breastfeeding / Lactation

Compatible

Patient Counseling & Practical Advice

How to Take:

Report visual changes immediately

What to Do if You Miss a Dose:

Take as soon as remembered

Recommended Monitoring & Lab Tests:

Baseline and annual eye exams, ECG

Emergency Medical Warning

When to Seek Urgent Medical Attention

Seek immediate emergency medical care (call emergency services or proceed to the nearest emergency department) if you experience signs of a life-threatening allergic reaction (anaphylaxis: facial, lip, tongue, or throat swelling causing airway obstruction), severe cutaneous blistering with skin peeling, sudden intense chest pain, or symptoms of overdose.

Emergency Safety Protocol: If an intentional or accidental overdose is suspected, contact your regional Poison Control Center or emergency services immediately. Do not induce vomiting unless strictly advised by emergency healthcare personnel.
Educational Sources & References

Content for Hydroxychloroquine was synthesized from standardized public health monographs, official pharmacopoeias, and health authorities:

  • Central Drugs Standard Control Organization (CDSCO) — National List of Essential Medicines
  • World Health Organization (WHO) — Model List of Essential Medicines
  • Indian Pharmacopoeia Commission (IPC) — Indian Pharmacopoeia Drug Monographs
  • National Health Service (NHS) — Medicines A to Z Clinical Guidelines
Published by: Medi Info Hub TeamLast Updated: 10/19/2026

The information provided on this website is for educational purposes only and is not intended as a substitute for professional medical advice, diagnosis, or treatment. Always seek the advice of a qualified healthcare provider with any questions you may have regarding a medical condition.